TITLE mglur
NEURON {
SUFFIX mglur
USEION glu READ gluo VALENCE -1
USEION ip3 WRITE iip3 VALENCE 1
NONSPECIFIC_CURRENT i
RANGE totalmGluR, GlumGluR, mGluR, r, i, iip3, K2
}
UNITS
{
(molar) = (1/liter)
(mM) = (millimolar)
(um) = (micron)
(mA) = (milliamp)
(mV) = (millivolt)
FARADAY = (faraday) (coulomb)
}
ASSIGNED {
gluo (mM)
vol (um3)
diam (um)
area (um2)
iip3 (mA/cm2)
i (mA/cm2)
}
STATE
{
mGluR (mM)
GlumGluR (mM)
}
PARAMETER {
totalmGluR = 30e-3 (mM)
K1 = 280 (/ms mM) : forward binding rate to receptor from Bhalla et al
K2 = 0.016 (/ms)
r = 0.2083e-3 (1): proportion of bindings that result in ip3 production
: given a clearance rate of 1/1000 if all mGluR are bound
: this gives steady-state ip3 of 100nm
}
BREAKPOINT {
SOLVE bindkin METHOD sparse
iip3 = -(1e-4) * r * (K2 * FARADAY * GlumGluR * vol/area)
i = -iip3
}
KINETIC bindkin {
~ gluo + mGluR <-> GlumGluR (K1, K2)
CONSERVE mGluR + GlumGluR = totalmGluR
}
INITIAL {
: changed basal gluo to 0
mGluR = totalmGluR : - K1*25e-6*totalmGluR/(K2 + K1*25e-6)
GlumGluR = 0 : K1*25e-6*totalmGluR/(K2 + K1*25e-6)
vol = area * diam
}